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5-氨基-1-甲基喹啉碘化物 98.0% | 42464-96-0


  • 产物称号
  • CasNo
  • 份子式
  • 份子量
  • 含量
  • 表面
  • 包装
  • 操纵
  • 5-氨基-1-甲基喹啉碘化物 98.0% | 42464-96-0
  • 42464-96-0
  • C10H11IN2
  • 286.11
  • 98.0%
  • 棕色-棕红色粉末
  • 1kg/包;25kg/桶
  • 增进老化肌肉的再生才能,增添满身瘦肉品德
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终产(chan)物头(tou)像(xiang)框

5-氨(an)基-1-甲(jia)基喹啉碘(dian)化物

国外英文微章(zhang)

5-Amino-1-methylquinolinium iodide(NNMTi)

日文被(bei)誉为

NNMTi

5-AMINO-1-METHYLQUINOLIN-1-IUM IODIDE

5-amino-1-methylquinolinium iodide

5-Amino-1-methylquinolin-1-iumiodide

1-methylquinolin-1-ium-5-amine;iodide

5-Amino-1-methyl-1-quinolinium Iodide

5-Amino-1-mq iodide

CAS No.

42464-96-0

份子式(shi)

C10H11IN2

份子量

286.11

含量

98.0%

表面(mian)能

浅棕(zong)色(se)-棕(zong)红碎末(mo)

包装(zhuang)箱

1kg/包;25kg/桶(tong)

储存本质

储放于封闭空(kong)间、空(kong)调、室内温度、无太阳光照射到的出所。

提示

本🐭(ben)公司的任何事物化合(he)物只(zhi)供出口国在(zai)合(he)理(li)合(he)法(fa)和非实(shi)用(yong)新型省份(fen)试过室和科(ke)技创新使用(yong)。不许小我或草本(ben)花卉使用(yong),不法(fa)分(fen)子使用(yong)不当者对在(zai)此产生的结杲负完🔯正(zheng)权利与义务。

1.结果先容

体(ti)(ti)細胞(bao)溶质酶烟酰胺 N-甲基改(gai)变酶 (NNMT) 已被新(xin)发明(ming)人,可(ke)(ke)其(qi)实(shi)食(shi)(shi)补 NAD+ 动物(wu)进(jin)行(xing)降(jiang)解需求(qiu)的(de)(de)(de)烟酰胺前体(ti)(ti)的(de)(de)(de)地(di)步(bu),是以在(zai)食(shi)(shi)补 NAD+ 挽回门(men)道和体(ti)(ti)細胞(bao)细胞(bao)产生(sheng)(sheng)率中(zhong)(zhong)起(qi)着特别重在(zai)的(de)(de)(de)作用(yong)(yong)。NNMT 在(zai)骨格肌(ji)(ji)(ji)(ji)中(zhong)(zhong)表达,跟肌(ji)(ji)(ji)(ji)結构的(de)(de)(de)朽(xiu)迈,其(qi)表达不断彰(zhang)显。重在(zai)的(de)(de)(de)是,NNMT 是肌(ji)(ji)(ji)(ji)消减症(zheng)遗传基因表达特性的(de)(de)(de)重在(zai)带来高(gao)斯模糊(hu),其(qi)苛刻表达可(ke)(ke)其(qi)实(shi)引(yin)致(zhi) NAD+ 地(di)步(bu)看不出(chu)起(qi)降(jiang),并亲(qin)自(zi)朽(xiu)迈而(er)呈现(xian)出(chu)来肌(ji)(ji)(ji)(ji)品格、的(de)(de)(de)强度和作用(yong)(y𓆏ong)与功郊(jiao)的(de)(de)(de)起(qi)降(jiang)。用(yong)(yong)小(xiao)份子 NNMT 按奈(nai)剂 (NNMTi) 医冶(ye)老龄人小(xiao)鼠(shu)需加(jia)强 muSC 的(de)(de)(de)增(zeng)(zeng)值、融会和降(jiang)解能力,导致(zhi)提升骨格肌(ji)(ji)(ji)(ji)的(de)(de)(de)作用(yong)(yong)与功郊(jiao)后能。在(zai)身体(ti)(ti)之外,操作与 muSC 很是近貌(mao)似(si) C2C12 体(ti)(ti)細胞(bao)也认定了近貌(mao)似(si)重大成(cheng)就(jiu),此中(zhong)(zhong) NNMTi 医冶(ye)增(zeng)(zeng)加(jia)了成(cheng)肌(ji)(ji)(ji)(ji)体(ti)(ti)細胞(bao)进(jin)行(xing)降(jiang)解并撑持 NAD+ 挽回门(men)道相(xiang)干体(ti)(ti)細胞(bao)细胞(bao)产生(sheng)(sheng)率物(wu)的(de)(de)(de)细胞(bao)产生(sheng)(sheng)率改(gai)变。

NNMTi 非种(zhong)(zhong)在背部(bu)(bu)(bu)肌肉骨骼肌老化(hua)(hua)测(ce)试发展中自私描(miao)写出(chu)(chu)(chu)的酶(mei),与复原(yuan) NAꦺD+ 径路毁伤、sirtuin1 化(hua)(hua)学活(huo)化(hua)(hua)义(yi)均教育和(he)背部(bu)(bu)(bu)肌肉干内部(bu)(bu)(bu)朽迈添置有关于。NNMT 非种(zhong)(zhong)分(fen)泌酶(mei),调控通用的甲(jia)基供体(ti) S-腺苷(gan)甲(jia)硫(liu)氨酸 (SAM) 催化(hua)(hua)反应(ying)烟酰胺 (NAM) 甲(jia)基化(hua)(hua),将内部(bu)(bu)(bu)的分(fen)泌的情(qing)形(xing)与甲(jia)基化(hua)(hua)义(yi)均教育和(he)内部(bu)(bu)(bu)内 NAD+ 层度(du)热(re)情(qing)接待(dai)上(shang)(shang)来。NNMT 在肝功(gong)能和(he)油脂内部(bu)(bu)(bu)结构和(he)以分(fen)泌需(xu)要添置为(wei)特色文化(hua)(hua)的病(bing)检(jian)的情(qing)形(xing)广州(zhou)中山大学量描(miao)写出(chu)(chu)(chu),目空一切某(mou)种(zhong)(zhong)油脂肝慢性病(bing)和(he)痛风。NNMT 出(chu)(chu)(chu)庭四种(zhong)(zhong)拆分(fen)发展,带有老辣到꧂熟我(wo)们人类胚(pei)胎干内部(bu)(bu)(bu)变化(hua)(hua)、肌一出(chu)(chu)(chu)生和(he)四种(zhong)(zhong)癌病(bing)中的上(shang)(shang)皮和(he)周围(wei)神经间质变化(hua)(hua)。NNMT 描(miao)写出(chu)(chu)(chu)以内部(bu)(bu)(bu)结构和(he)环境特男(nan)男(nan)的体(ti)例食补,而非经过发展覆盖全国(guo)现实存在的食补形(xing)势食补。

2.一大特(te)色

 (1)纯净(jing)度(du)(du)就(jiu)越高:NNMTi通(tong)过速度(du)(du)特制主产🔴地生(sheng)产工(gong)艺就(jiu)可(ke)以或者是选取(qu)高纯净(jing)度(du)(du)的(de)货物,高纯净(jing)度(du)(du)代表(biao)着更(geng)佳的(de)动(dong)物操控度(du)(du)。

(2)靶点性:NNMTi特别(bie)对于NNMT酶(mei),都可以我以为要用(yong)抑制其(qi)活(huo)性氧,然后直接影响(xiang)烟(yan)酰(xian)胺的⛦基础代谢(xie)好(hao)项目。

(3)没变性:NNMTi具备(bei)条(tiao)件典范的(de)没变性,在差另一个要素和(he)存贮要素下都🐻能始终坚持其活🐼性酶(mei)类和(he)最终结果(guo)。

(4)建(jian)立前景:为了NNMTi的几种特证,建(jian)立🌳诬陷广(guang)泛(fan)存眷,具备广(guang)泛(fan)的研究(ji🃏u)讨论和控制前景。

3.使(shi)用基本概念

NNMTi (CAS 42464-96-0) 有的(de)(de)(de)是种(zhong)烟酰胺(an) N-甲(jia)基更改(gai)酶(mei) (NNMT) 按(an)(an)耐剂(ji),有的(de)(de)(de)是种(zhong)有效果(guo)的(de)(de)(de)烟酰胺(an) N -甲(jia)基更改(gai)酶(mei) (NNMT) 的(de)(de)(de)按(an)(an)耐剂(ji) (IC50=1.2 μM),可(ke)提(ti)升(sheng)成肌生殖(zhi)癌内(nei)(nei)(nei)部(bu)溶(rong)解(jie)。NNMTi 必选择性(xing)地(di)(di)取(qu)(qu)得联(lian)(lian)系 NNMT 底物(wu)(wu)取(qu)(qu)得联(lian)(lian)系位点残基。NNMTi 能提(ti)升(sheng)身(shen)体成肌生殖(zhi)癌内(nei)(nei)(nei)部(bu)溶(rong)解(jie),继续加强年(nian)龄较大的(de)(de)(de)小鼠背部(bu)相(xiang)关(guan)肌干生殖🍃(zhi)癌内(nei)(nei)(nei)部(bu)融(rong)会和重(zhong)复(fu)就(jiu)能。NNMT 有的(de)(de)(de)是种(zhong)基石的(de)(de)(de)生殖(zhi)癌内(nei)(nei)(nei)部(bu)溶(rong)质海(hai)洋怪物(wu)(wu)流(liu)量(liang)转化酶(mei),可(ke)促使(shi)内(nei)(nei)(nei)源性(xing)和外源性(xing)外地(di)(di)人海(hai)洋怪物(wu)(wu)的(de)(de)(de) N-甲(jia)基化。与(yu)纯确实鸡(ji)肉食用编辑借喻,NNMTi 医好与(yu)鸡(ji)肉食用编辑相(xiang)取(qu)(qu)得联(lian)(lian)系要加速(su)升(sheng)级重(zhong)量(liang)乳(ru)(ru)酸(suan)核(he)减(jian)(jian)、曾加身(shen)上鸡(ji)肉品质与(yu)重(zhong)量(liang)比、核(he)减(jian)(jian)肝部(bu)附睾颜色乳(ru)(ru)酸(suan)构建权重(zhong)、核(he)减(jian)(jian)肝部(bu)乳(ru)(ru)酸(suan)堆积作用、升(sheng)级肝部(bu)乳(ru)(ru)酸(suan)男(nan)变女(nv)。与(yu)此同时NNMTi 都可(ke)以如(ru)(ru)果(guo)你曾加气血并提(ti)升(sheng)老化测试背部(bu)相(xiang)关(guan)肌的(de)(de)(de)重(zhong)复(fu)就(jiu)能,这都可(ke)以如(ru)(ru)果(guo)你这样有利于医好背部(bu)相(xiang)关(guan)肌核(he)减(jian)(jian)症。

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